Basic Information
ID: ALA4056010
Type: Binding
Description: Displacement of (P)-1-(30-chloro-2-fluoro-5,50-dimethoxy-[1,10biphenyl]-4-yl)-N-(isoxazol-3-yl)-2-oxo-1,2-dihydroquinoline-6-sulfonamide[50-methoxy-C3H3] from human NaV1.7 expressed in HEK293 cell membranes incubated for 1 hr by beta counting method
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4056010
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 510.54 | 5.49 | 5.49 |
| 500.91 | 5.02 | 5.02 |
| 484.46 | 4.50 | 4.50 |
| 467.45 | 3.76 | 3.76 |