Basic Information
ID: ALA4058264
Type: Binding
Description: Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD4 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Bromodomain-containing protein 4(ALA1163125)
Document: ALA4052791
Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD4 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4058264
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 392.50 | 3.16 | 3.16 |
| 330.43 | 1.81 | 1.81 |
| 432.57 | 4.12 | 4.12 |
| 432.57 | 4.12 | 4.12 |
| 302.38 | 1.03 | 1.03 |
| 418.54 | 3.81 | 3.81 |
| 288.35 | 0.69 | 0.69 |