Assay Report Card

Basic Information

ID: ALA4119867

Type: Binding

Description: Binding affinity to N-terminally GST-tagged wild type human DLK (1 to 520 residues) expressed in sf21 insect cells using N-terminally His-tagged MKK4 K131M as substrate after 60 mins in presence of ATP by TR-FRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
379.513.893.89
415.414.044.04
433.484.604.60
399.934.244.24
383.473.723.72
409.463.713.71
375.903.343.34
355.492.992.99
371.492.702.70
393.413.323.32
409.463.423.42
407.443.173.17
405.452.752.75
369.472.162.16
419.453.003.00
389.453.093.09
433.483.393.39
423.443.053.05
447.383.153.15
435.452.882.88
421.473.423.42
379.392.132.13
437.472.362.36
395.392.012.01
447.513.783.78
421.473.253.25
409.463.153.15
393.412.612.61