Basic Information
ID: ALA4121728
Type: Binding
Description: Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrate addition measured after 120 mins by fluorescence polarization assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4121728
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 392.44 | 4.00 | 4.00 |
| 328.37 | 4.68 | 4.68 |
| 314.34 | 4.60 | 4.60 |
| 370.45 | 5.79 | 5.79 |
| 342.40 | 5.16 | 5.16 |
| 382.46 | 6.25 | 6.25 |
| 306.37 | 4.59 | 4.59 |
| 370.46 | 4.06 | 4.06 |
| 263.26 | 2.80 | 2.80 |
| 370.46 | 4.06 | 4.06 |
| 304.35 | 3.32 | 3.32 |
| 456.55 | 4.02 | 4.02 |
| 406.44 | 6.39 | 6.39 |
| 321.34 | 3.59 | 3.59 |
| 411.51 | 5.66 | 5.66 |
| 396.88 | 4.77 | 4.77 |
| 498.63 | 5.14 | 5.14 |
| 366.42 | 4.65 | 4.65 |
| 238.25 | 2.93 | 2.93 |
| 441.54 | 3.68 | 3.68 |
| 424.55 | 5.72 | 5.72 |
| 237.26 | 2.33 | 2.33 |
| 331.38 | 4.46 | 4.46 |
| 438.53 | 4.79 | 4.79 |
| 441.54 | 3.68 | 3.68 |
| 356.43 | 5.72 | 5.72 |
| 367.41 | 5.25 | 5.25 |
| 426.52 | 4.14 | 4.14 |
| 330.39 | 3.86 | 3.86 |
| 456.55 | 4.02 | 4.02 |
| 439.56 | 6.44 | 6.44 |
| 362.43 | 4.12 | 4.12 |
| 391.45 | 3.40 | 3.40 |
| 380.42 | 4.26 | 4.26 |
| 406.47 | 3.37 | 3.37 |
| 449.48 | 6.67 | 6.67 |
| 406.47 | 3.37 | 3.37 |
| 320.39 | 4.89 | 4.89 |
| 450.59 | 6.03 | 6.03 |
| 328.37 | 4.90 | 4.90 |
| 480.61 | 5.91 | 5.91 |
| 411.51 | 5.66 | 5.66 |
| 396.45 | 4.66 | 4.66 |
| 456.55 | 4.02 | 4.02 |
| 465.48 | 6.55 | 6.55 |
| 426.52 | 4.14 | 4.14 |
| 397.48 | 5.36 | 5.36 |
| 320.35 | 2.99 | 2.99 |
| 305.34 | 3.92 | 3.92 |
| 381.41 | 4.86 | 4.86 |
| 343.39 | 4.00 | 4.00 |
| 349.39 | 3.68 | 3.68 |
| 363.42 | 4.72 | 4.72 |
| 338.37 | 3.87 | 3.87 |
| 468.60 | 5.26 | 5.26 |
| 384.41 | 4.79 | 4.79 |
| 408.51 | 4.91 | 4.91 |
| 380.45 | 4.96 | 4.96 |
| 420.52 | 5.72 | 5.72 |
| 473.58 | 7.45 | 7.45 |
| 405.46 | 5.79 | 5.79 |
| 426.52 | 4.14 | 4.14 |