Basic Information
ID: ALA4122972
Type: Binding
Description: Inhibition of KDM5A (M1 to L801 residues) PHD2/3 deletion mutant (unknown origin) demethylation activity preincubated for 10 mins followed by peptide addition measured after 3 mins by MALDI-TOF-MS analysis
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4122972
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 645.32 | 6.94 | 6.94 |
| 307.40 | -0.32 | -0.32 |
| 379.50 | 5.34 | 5.34 |
| 773.23 | 6.69 | 6.69 |
| 521.44 | 5.48 | 5.48 |