Basic Information
ID: ALA4122985
Type: Binding
Description: Mixed type inhibition of KDM5A (L88 to G353 residues) ARID/PHD1/2/3 deletion mutant (unknown origin) demethylation activity using H3(1-21)K4me3 peptide as substrate measured every 30 seconds over 25 mins by formaldehyde dehydrogenase coupled activity assay based Lineweaver-Burk plot analysis
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4122985
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 521.44 | 5.48 | 5.48 |