Assay Report Card

Basic Information

ID: ALA4134888

Type: Binding

Description: Inhibition of human FLAG-tagged TRPM2 expressed in HEK293 cells assessed as reduction in ADPR-induced intracellular calcium flux at 2 uM treated for 6 hrs followed by compound washout measured within 5 mins by whole cell patch clamp electrophysiology method

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
428.615.545.54