Basic Information
ID: ALA4136963
Type: Binding
Description: Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine nucleotide exchange activity using BODIPY-labeled GDP loaded Rap1A by fluorescence assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4136963
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 351.01 | 3.65 | 3.65 |
| 367.08 | 4.45 | 4.45 |
| 351.01 | 3.65 | 3.65 |
| 367.08 | 4.45 | 4.45 |