Basic Information
ID: ALA4137466
Type: Binding
Description: Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4137466
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 244.21 | -3.17 | -3.17 |
| 490.65 | 3.87 | 3.87 |
| 228.21 | -2.14 | -2.14 |
| 509.74 | 5.84 | 5.84 |
| 461.53 | 5.65 | 5.65 |
| 546.71 | 5.02 | 5.02 |
| 494.71 | 5.65 | 5.65 |
| 480.70 | 5.66 | 5.66 |
| 521.71 | 4.98 | 4.98 |
| 492.66 | 5.44 | 5.44 |
| 478.64 | 4.01 | 4.01 |
| 508.75 | 6.44 | 6.44 |
| 504.68 | 5.72 | 5.72 |
| 491.64 | 3.97 | 3.97 |
| 496.70 | 3.37 | 3.37 |
| 464.61 | 4.84 | 4.84 |
| 412.58 | 3.92 | 3.92 |
| 489.62 | 4.75 | 4.75 |
| 475.64 | 4.68 | 4.68 |
| 482.67 | 4.85 | 4.85 |
| 540.71 | 6.54 | 6.54 |
| 466.55 | 4.63 | 4.63 |
| 521.71 | 4.94 | 4.94 |
| 482.67 | 4.51 | 4.51 |
| 478.64 | 4.01 | 4.01 |
| 478.64 | 5.18 | 5.18 |
| 477.65 | 4.92 | 4.92 |
| 479.63 | 4.58 | 4.58 |
| 506.69 | 5.96 | 5.96 |
| 428.58 | 3.62 | 3.62 |
| 520.72 | 6.22 | 6.22 |
| 464.61 | 4.87 | 4.87 |
| 478.68 | 5.57 | 5.57 |
| 514.67 | 6.03 | 6.03 |
| 474.65 | 5.28 | 5.28 |
| 494.64 | 4.37 | 4.37 |
| 488.68 | 5.59 | 5.59 |
| 518.70 | 5.97 | 5.97 |
| 480.65 | 4.42 | 4.42 |