Basic Information
ID: ALA4139703
Type: Binding
Description: Inhibition of N-terminal His6-tagged KAT8 catalytic domain (125 to 458 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGKGGKGLGKGGAKRHRK-NH2 as substrate after 5 mins in presence of Ac-CoA by fluorescence assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4139703
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 125.15 | 1.28 | 1.28 |
| 127.57 | 1.92 | 1.92 |
| 111.12 | 1.41 | 1.41 |
| 143.19 | 2.42 | 2.42 |
| 109.13 | 0.97 | 0.97 |
| 173.17 | 2.75 | 2.75 |
| 108.14 | 0.97 | 0.97 |
| 159.19 | 2.13 | 2.13 |
| 145.16 | 1.94 | 1.94 |
| 189.17 | 2.45 | 2.45 |
| 144.60 | 0.97 | 0.97 |
| 160.18 | 1.52 | 1.52 |
| 223.70 | 2.61 | 2.61 |
| 215.25 | 2.89 | 2.89 |
| 277.32 | 3.73 | 3.73 |
| 213.50 | 2.28 | 2.28 |
| 223.25 | 1.67 | 1.67 |
| 187.20 | 1.64 | 1.64 |
| 313.38 | 3.65 | 3.65 |
| 174.63 | 0.98 | 0.98 |
| 201.22 | 2.35 | 2.35 |
| 168.20 | 2.29 | 2.29 |
| 201.22 | 2.50 | 2.50 |
| 189.21 | 2.14 | 2.14 |
| 313.44 | 5.62 | 5.62 |
| 237.28 | 1.92 | 1.92 |
| 249.31 | 4.00 | 4.00 |
| 173.21 | 1.91 | 1.91 |
| 209.68 | 2.00 | 2.00 |
| 162.59 | 1.11 | 1.11 |
| 209.68 | 2.43 | 2.43 |