Basic Information
ID: ALA4141001
Type: Binding
Description: Inhibition of recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)-D-Arg-NH2 as substrate pretreated for 15 mins followed by substrate addition measured at 5 mins interval for 120 mins by fluorescence assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4141001
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 685.90 | 1.47 | 1.47 |
| 1174.44 | ||
| 1188.47 | ||
| 965.16 | 0.26 | 0.26 |
| 1134.43 | ||
| 965.16 | 0.26 | 0.26 |
| 945.17 | 0.15 | 0.15 |
| 959.20 | 0.54 | 0.54 |
| 973.22 | 0.79 | 0.79 |