ID: ALA4144986
Type: Binding
Description: Inverse agonist activity at biotinylated RORgammat LBD (unknown origin) assessed as inhibition of N-(2-chloro-6-fluorobenzyl)-N-((2'-methoxy-[1,1'-biphenyl]-4-yl)methyl)benzenesulfonamide-induced co-activator SRC1 peptide recruitment after 1 hr by dual FRET based LANCE assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4144986
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
490.61 | 5.02 | 5.02 |
481.92 | 6.00 | 6.00 |
611.69 | 6.02 | 6.02 |
653.77 | 7.05 | 7.05 |
413.46 | 4.80 | 4.80 |
504.63 | 5.32 | 5.32 |
447.48 | 5.35 | 5.35 |
663.20 | 7.83 | 7.83 |