Assay Report Card

Basic Information

ID: ALA4144986

Type: Binding

Description: Inverse agonist activity at biotinylated RORgammat LBD (unknown origin) assessed as inhibition of N-(2-chloro-6-fluorobenzyl)-N-((2'-methoxy-[1,1'-biphenyl]-4-yl)methyl)benzenesulfonamide-induced co-activator SRC1 peptide recruitment after 1 hr by dual FRET based LANCE assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
490.615.025.02
481.926.006.00
611.696.026.02
653.777.057.05
413.464.804.80
504.635.325.32
447.485.355.35
663.207.837.83