Basic Information
ID: ALA4145323
Type: Functional
Description: Antagonist activity at human KOR expressed in CHO cell membranes assessed as inhibition of U50488-induced [35S]-GTPgammaS binding preincubated for 5 mins followed by U50488 and [35S]-GTPgammaS addition measured after 80 mins
Organism: Homo sapiens
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA4145323
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 621.74 | 2.35 | 2.35 |
| 661.80 | 3.82 | 3.82 |
| 1385.63 | ||
| 340.38 | 1.30 | 1.30 |