Basic Information
ID: ALA4148663
Type: Binding
Description: Displacement of [3H]DTG from sigma-2 receptor in Sprague-Dawley rat liver membranes at 1 uM after 120 mins in presence of (+)-pentazocine by microbeta scintillation counting method relative to control
Organism: Rattus norvegicus
Strain: Sprague-Dawley
Tissue: Liver
Subcellular Fraction: Membrane
Activity Charts
Bioactivity
Activity Types for Assay ALA4148663
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 399.53 | 4.28 | 4.28 |
| 458.90 | 3.42 | 3.42 |
| 439.51 | 2.88 | 2.88 |
| 445.51 | 3.37 | 3.37 |
| 415.53 | 3.98 | 3.98 |
| 397.52 | 4.43 | 4.43 |
| 472.93 | 3.81 | 3.81 |
| 385.46 | 3.35 | 3.35 |
| 373.45 | 2.81 | 2.81 |
| 444.88 | 3.03 | 3.03 |
| 453.54 | 3.27 | 3.27 |
| 371.48 | 3.50 | 3.50 |
| 413.51 | 4.13 | 4.13 |
| 387.48 | 3.20 | 3.20 |
| 371.43 | 2.96 | 2.96 |
| 369.46 | 3.65 | 3.65 |