Assay Report Card

Basic Information

ID: ALA4150992

Type: Binding

Description: Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cells after 30 mins by fluorescence polarization assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
457.545.445.44
471.505.475.47
457.545.065.06
471.505.475.47
459.555.475.47
457.545.675.67
437.506.166.16
483.534.794.79
457.545.365.36
471.505.475.47
471.445.205.20
445.535.535.53
471.576.066.06
439.485.325.32
457.545.065.06
454.494.734.73
454.494.734.73
513.526.026.02
459.555.705.70
435.495.925.92
417.474.494.49
443.514.674.67
483.535.345.34
443.515.055.05
431.504.974.97
453.515.335.33
417.474.494.49
471.505.475.47
445.535.305.30
487.955.985.98
454.494.734.73