ID: ALA4150992
Type: Binding
Description: Inhibition of FAM-labeled ZBA248 binding to recombinant human BRD4 bromodomain 1 (44 to 168 residues) expressed in Rosetta2 Escherichia coli DE3 cells after 30 mins by fluorescence polarization assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4150992
Ki
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
457.54 | 5.44 | 5.44 |
471.50 | 5.47 | 5.47 |
457.54 | 5.06 | 5.06 |
471.50 | 5.47 | 5.47 |
459.55 | 5.47 | 5.47 |
457.54 | 5.67 | 5.67 |
437.50 | 6.16 | 6.16 |
483.53 | 4.79 | 4.79 |
457.54 | 5.36 | 5.36 |
471.50 | 5.47 | 5.47 |
471.44 | 5.20 | 5.20 |
445.53 | 5.53 | 5.53 |
471.57 | 6.06 | 6.06 |
439.48 | 5.32 | 5.32 |
457.54 | 5.06 | 5.06 |
454.49 | 4.73 | 4.73 |
454.49 | 4.73 | 4.73 |
513.52 | 6.02 | 6.02 |
459.55 | 5.70 | 5.70 |
435.49 | 5.92 | 5.92 |
417.47 | 4.49 | 4.49 |
443.51 | 4.67 | 4.67 |
483.53 | 5.34 | 5.34 |
443.51 | 5.05 | 5.05 |
431.50 | 4.97 | 4.97 |
453.51 | 5.33 | 5.33 |
417.47 | 4.49 | 4.49 |
471.50 | 5.47 | 5.47 |
445.53 | 5.30 | 5.30 |
487.95 | 5.98 | 5.98 |
454.49 | 4.73 | 4.73 |