Assay Report Card

Basic Information

ID: ALA4153629

Type: Binding

Description: Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) at 33 uM preincubated for 15 mins followed by biotin tagged H3 peptide ( 1 to 23 residues) and [3H]-Ac-CoA addition and measured after 60 mins by radioactive acetylation assay

Organism: Saccharomyces cerevisiae

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
534.497.007.00
473.534.674.67
414.464.464.46
444.375.135.13
496.385.875.87