Basic Information
ID: ALA4154872
Type: Binding
Description: Inhibition of His6-tagged human CREBBP (R1081 to G1197 residues) expressed in Escherichia coli BL21(DE3) using biotinylated-H4KAc4 as substrate by AlphaScreen assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4154872
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 509.05 | 5.48 | 5.48 |
| 338.34 | 4.17 | 4.17 |
| 320.35 | 4.03 | 4.03 |
| 300.36 | 3.70 | 3.70 |
| 326.40 | 3.87 | 3.87 |
| 298.34 | 3.46 | 3.46 |
| 411.50 | 3.18 | 3.18 |