Assay Report Card

Basic Information

ID: ALA4154879

Type: Binding

Description: Binding affinity to His6-tagged human EP300 (A1040 to G1161 residues) expressed in Escherichia coli BL21(DE3) assessed as change in melting temperature at 200 uM by SYPRO orange dye based fluorescence assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
457.005.535.53
338.344.174.17
320.354.034.03
300.363.703.70
326.403.873.87
298.343.463.46
411.503.183.18