Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincuba...

Basic Information

ID: ALA4155949

Type: Functional

Description: Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincubated for 60 mins followed by delta9-THC addition for 90 mins measured for 1 sec by luminescence assay

Format: BAO_0000219

Organism: Homo sapiens

Cell type: CHO

Target:  N-arachidonyl glycine receptor(ALA2384898)

Document:  ALA4152303

Antagonist activity at recombinant human GPR18 expressed in CHO cells assessed as inhibition of delta9-THC-induced beta-arrestin recruitment preincubated for 60 mins followed by delta9-THC addition for 90 mins measured for 1 sec by luminescence assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
452.945.825.82
485.056.426.42
345.814.244.24
344.823.263.26
368.434.084.08
464.636.006.00
428.944.864.86
414.914.474.47
513.846.446.44
471.026.036.03
358.854.114.11
464.635.945.94
364.473.983.98
463.006.336.33
434.955.685.68
429.344.704.70
471.026.036.03
370.864.204.20
378.504.374.37
499.086.816.81
341.803.263.26
469.396.336.33
471.026.036.03
478.666.506.50
442.975.255.25
364.474.254.25
361.884.414.41
448.985.995.99
372.884.454.45
450.605.695.69
457.005.645.64
370.864.204.20
448.985.725.72