Basic Information
ID: ALA4181270
Type: Binding
Description: Antagonist activity at recombinant full length EPAC2 (unknown origin) assessed as inhibition of cAMP-mediated Rap1b-BODIPY GDP nucleotide exchange activity
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4181270
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 330.78 | 3.80 | 3.80 |
| 351.01 | 3.65 | 3.65 |
| 400.31 | 6.22 | 6.22 |
| 415.32 | 5.15 | 5.15 |
| 441.38 | 6.20 | 6.20 |
| 407.82 | 5.83 | 5.83 |
| 352.61 | 4.82 | 4.82 |
| 378.21 | 4.18 | 4.18 |
| 394.26 | 5.83 | 5.83 |
| 357.82 | 4.95 | 4.95 |
| 376.20 | 3.95 | 3.95 |
| 374.27 | 5.47 | 5.47 |
| 407.82 | 5.83 | 5.83 |
| 372.26 | 5.05 | 5.05 |
| 357.82 | 4.95 | 4.95 |
| 368.22 | 5.32 | 5.32 |
| 352.61 | 4.82 | 4.82 |
| 359.35 | 4.58 | 4.58 |
| 339.83 | 4.81 | 4.81 |
| 408.72 | 6.12 | 6.12 |
| 369.21 | 4.72 | 4.72 |
| 407.82 | 5.83 | 5.83 |
| 402.16 | 5.07 | 5.07 |
| 417.30 | 4.00 | 4.00 |