Assay Report Card

Basic Information

ID: ALA4182256

Type: Binding

Description: Inhibition of recombinant human BRD2 bromodomain 2 (342 to 460 residues) using biotin labeled peptide substrate preincubated for 15 mins followed by substrate addition measured after 1 hr by TR-FRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
457.005.535.53
434.926.006.00
355.444.004.00
372.494.744.74
355.444.004.00
356.424.274.27
356.424.274.27
372.494.744.74