Reversible inhibition of 20s constitutive proteasome beta5 chymotrypsin-like activity in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate...

Basic Information

ID: ALA4185014

Type: Binding

Description: Reversible inhibition of 20s constitutive proteasome beta5 chymotrypsin-like activity in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate at 50 uM preincubated for 30 mins followed by compound dilution measured after 30 mins by fluorescence assay

Format: BAO_0000219

Organism: Homo sapiens

Target:  Proteasome Macropain subunit MB1(ALA4662)

Document:  ALA4184119

Reversible inhibition of 20s constitutive proteasome beta5 chymotrypsin-like activity in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate at 50 uM preincubated for 30 mins followed by compound dilution measured after 30 mins by fluorescence assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
340.402.972.97