Assay Report Card

Basic Information

ID: ALA4187420

Type: Binding

Description: Inhibition of N-terminal GST-HIS6 fusion protein tagged human CDK7 (M1 to F346 residues)/N-terminal HIS6-tagged human Cyclin-H (M1 to L323 residues)/N-terminal HIS6-tagged human MAT1 (M1 to S306 residues) expressed in Sf9 cells at 1 uM using RB-CTF substrate and ATP incubated for 1 hr by fluorescent polarization assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
483.534.834.83
487.494.584.58
407.485.295.29
469.504.444.44
469.504.444.44
472.534.004.00
469.504.444.44
425.475.435.43
457.514.294.29
490.524.134.13