Assay Report Card

Basic Information

ID: ALA4187422

Type: Binding

Description: Inhibition of human full length CDK2 (M1 to L298 residues)/human full length Cyclin-A2 (M1 to L432 residues) expressed in Sf9 cells at 1 uM using TAMRA-histone H1-derived peptide substrate and ATP incubated for 1 hr by fluorescent polarization assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
483.534.834.83
487.494.584.58
407.485.295.29
469.504.444.44
469.504.444.44
472.534.004.00
469.504.444.44
425.475.435.43
457.514.294.29
490.524.134.13