Assay Report Card

Basic Information

ID: ALA4189068

Type: Binding

Description: Inhibition of wild type recombinant human histone lysine methyltransferase G9a (913 to 1193 residues) expressed in Escherichia coli Rosetta BL21 DE3 PlysS assessed as zinc ions ejection from Cys4-Zn finger at 100 uM by FluoZin-3 based fluorescence assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
78.14-0.01-0.01
77.15-0.13-0.13
116.08-0.40-0.40
189.07
274.18
208.222.462.46
158.161.621.62
296.553.623.62
171.271.541.54
188.94
240.442.062.06
220.323.283.28
307.33-2.21-2.21
178.14-0.25-0.25
509.745.845.84
225.210.290.29
312.13
191.52
235.97
302.19