Basic Information
ID: ALA4189162
Type: Binding
Description: Agonist activity at human N-terminal alphaHis-SUMO-tagged ERRgamma-LBD (229 to 458 residues) expressed in Escherichia coli BL21 gold (DE3) cells assessed as decrease in RIP140 peptide recruitment after 2 hrs by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4189162
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 282.34 | 3.28 | 3.28 |
| 193.25 | 1.78 | 1.78 |
| 207.27 | 2.17 | 2.17 |
| 236.31 | 1.46 | 1.46 |
| 365.39 | 4.68 | 4.68 |
| 310.40 | 3.84 | 3.84 |
| 297.40 | 3.66 | 3.66 |
| 326.40 | 3.06 | 3.06 |
| 282.39 | 3.35 | 3.35 |
| 320.44 | 4.44 | 4.44 |
| 295.38 | 4.34 | 4.34 |
| 234.30 | 1.22 | 1.22 |
| 298.39 | 3.06 | 3.06 |
| 340.47 | 3.99 | 3.99 |
| 296.37 | 3.45 | 3.45 |
| 320.44 | 4.44 | 4.44 |
| 297.40 | 3.66 | 3.66 |
| 430.55 | 5.29 | 5.29 |
| 312.41 | 3.21 | 3.21 |
| 311.43 | 4.00 | 4.00 |
| 315.39 | 3.80 | 3.80 |
| 310.40 | 2.96 | 2.96 |
| 311.43 | 3.45 | 3.45 |
| 311.43 | 3.97 | 3.97 |
| 258.25 | 2.30 | 2.30 |
| 342.40 | 3.57 | 3.57 |
| 296.37 | 3.45 | 3.45 |
| 322.41 | 3.53 | 3.53 |
| 315.39 | 3.80 | 3.80 |
| 324.38 | 3.45 | 3.45 |
| 290.32 | 3.31 | 3.31 |
| 340.47 | 3.99 | 3.99 |
| 320.44 | 4.44 | 4.44 |
| 326.44 | 3.60 | 3.60 |
| 374.48 | 4.72 | 4.72 |
| 284.36 | 4.33 | 4.33 |
| 334.42 | 4.64 | 4.64 |
| 354.45 | 3.62 | 3.62 |
| 333.45 | 3.21 | 3.21 |
| 376.29 | 4.42 | 4.42 |
| 298.39 | 3.06 | 3.06 |
| 248.33 | 1.61 | 1.61 |
| 311.43 | 3.97 | 3.97 |
| 387.52 | 5.64 | 5.64 |
| 250.30 | 0.45 | 0.45 |
| 311.43 | 3.59 | 3.59 |
| 239.27 | 2.79 | 2.79 |
| 326.40 | 2.20 | 2.20 |
| 296.37 | 3.45 | 3.45 |
| 430.55 | 5.29 | 5.29 |
| 296.41 | 3.54 | 3.54 |
| 346.86 | 3.86 | 3.86 |
| 320.19 | 3.13 | 3.13 |
| 283.37 | 3.62 | 3.62 |
| 310.40 | 3.76 | 3.76 |
| 280.37 | 3.75 | 3.75 |
| 373.50 | 5.33 | 5.33 |
| 340.47 | 3.73 | 3.73 |
| 313.40 | 3.37 | 3.37 |
| 317.39 | 4.03 | 4.03 |
| 312.37 | 3.65 | 3.65 |
| 303.45 | 3.19 | 3.19 |
| 327.42 | 3.67 | 3.67 |
| 297.40 | 2.93 | 2.93 |
| 303.45 | 3.19 | 3.19 |
| 303.43 | 3.72 | 3.72 |
| 326.40 | 2.74 | 2.74 |
| 340.47 | 3.99 | 3.99 |
| 312.41 | 3.53 | 3.53 |
| 387.52 | 5.64 | 5.64 |
| 374.48 | 4.72 | 4.72 |
| 331.84 | 4.32 | 4.32 |
| 284.36 | 2.80 | 2.80 |
| 387.52 | 5.64 | 5.64 |
| 391.31 | 3.97 | 3.97 |
| 311.43 | 4.05 | 4.05 |
| 280.37 | 4.59 | 4.59 |
| 337.42 | 3.11 | 3.11 |