Assay Report Card

Basic Information

ID: ALA4189167

Type: Binding

Description: Partial agonist activity at human N-terminal alphaHis-SUMO-tagged ERRgamma-LBD (229 to 458 residues) expressed in Escherichia coli BL21 gold (DE3) cells assessed as decrease in RIP140 peptide recruitment after 2 hrs by TR-FRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
312.373.163.16
340.473.853.85
298.393.123.12
281.403.963.96
374.484.394.39
312.413.243.24
323.402.852.85
337.423.713.71
283.332.222.22