ID: ALA4189167
Type: Binding
Description: Partial agonist activity at human N-terminal alphaHis-SUMO-tagged ERRgamma-LBD (229 to 458 residues) expressed in Escherichia coli BL21 gold (DE3) cells assessed as decrease in RIP140 peptide recruitment after 2 hrs by TR-FRET assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4189167
EC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
312.37 | 3.16 | 3.16 |
340.47 | 3.85 | 3.85 |
298.39 | 3.12 | 3.12 |
281.40 | 3.96 | 3.96 |
374.48 | 4.39 | 4.39 |
312.41 | 3.24 | 3.24 |
323.40 | 2.85 | 2.85 |
337.42 | 3.71 | 3.71 |
283.33 | 2.22 | 2.22 |