Basic Information
ID: ALA4189551
Type: Binding
Description: Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate after 60 mins by caliper assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4189551
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 146.15 | 1.34 | 1.34 |
| 133.15 | 1.15 | 1.15 |
| 194.23 | 2.25 | 2.25 |
| 162.19 | 1.91 | 1.91 |
| 395.47 | 4.20 | 4.20 |
| 161.16 | 0.66 | 0.66 |
| 249.27 | 2.47 | 2.47 |
| 395.42 | 4.05 | 4.05 |
| 289.34 | 2.72 | 2.72 |
| 213.24 | 1.92 | 1.92 |
| 248.29 | 3.41 | 3.41 |
| 248.29 | 3.12 | 3.12 |
| 166.61 | 2.52 | 2.52 |
| 164.21 | 1.51 | 1.51 |
| 152.58 | 2.22 | 2.22 |
| 235.25 | 2.27 | 2.27 |
| 339.40 | 4.03 | 4.03 |
| 381.44 | 4.16 | 4.16 |
| 395.47 | 4.50 | 4.50 |
| 197.03 | 2.33 | 2.33 |
| 234.26 | 2.88 | 2.88 |
| 237.26 | 2.33 | 2.33 |
| 204.30 | 2.53 | 2.53 |
| 382.43 | 3.58 | 3.58 |
| 409.49 | 4.59 | 4.59 |
| 317.40 | 3.50 | 3.50 |
| 369.43 | 4.04 | 4.04 |
| 251.29 | 3.03 | 3.03 |
| 185.23 | 2.24 | 2.24 |
| 233.27 | 3.71 | 3.71 |
| 382.43 | 3.55 | 3.55 |
| 339.40 | 4.03 | 4.03 |
| 234.26 | 3.11 | 3.11 |
| 427.48 | 4.54 | 4.54 |
| 179.24 | 1.26 | 1.26 |
| 382.43 | 3.58 | 3.58 |
| 381.44 | 4.18 | 4.18 |
| 325.38 | 4.02 | 4.02 |
| 382.43 | 3.55 | 3.55 |
| 195.22 | 2.62 | 2.62 |
| 423.48 | 4.42 | 4.42 |
| 351.41 | 4.17 | 4.17 |
| 324.39 | 4.88 | 4.88 |
| 194.28 | 1.82 | 1.82 |
| 248.29 | 3.12 | 3.12 |
| 146.19 | 1.76 | 1.76 |
| 381.44 | 4.16 | 4.16 |
| 203.29 | 2.39 | 2.39 |
| 317.40 | 3.50 | 3.50 |
| 311.35 | 3.96 | 3.96 |
| 245.28 | 3.78 | 3.78 |
| 263.10 | 2.51 | 2.51 |