ID: ALA4189951
Type: Binding
Description: Displacement of MRS4174 from human P2Y14R expressed in CHO cells preincubated for 30 mins followed by MRS4174 addition measured after 30 mins by flow cytometric method
Organism: Homo sapiens
Cell type: CHO
Bioactivity
Activity Types for Assay ALA4189951
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
475.51 | 7.36 | 7.36 |
513.55 | 4.79 | 4.79 |
488.40 | 4.68 | 4.68 |
349.27 | 3.36 | 3.36 |
637.66 | 5.18 | 5.18 |
565.60 | 4.40 | 4.40 |
499.45 | 3.99 | 3.99 |
332.28 | 4.93 | 4.93 |
627.64 | 6.07 | 6.07 |
613.66 | 6.43 | 6.43 |
657.67 | 5.56 | 5.56 |
515.52 | 4.46 | 4.46 |
516.53 | 5.27 | 5.27 |
515.52 | 4.46 | 4.46 |
475.36 | 3.81 | 3.81 |
530.48 | 5.85 | 5.85 |
476.42 | 3.90 | 3.90 |
532.53 | 5.33 | 5.33 |
663.70 | 5.62 | 5.62 |
537.54 | 3.62 | 3.62 |
665.72 | 5.96 | 5.96 |
543.55 | 4.01 | 4.01 |
553.59 | 4.42 | 4.42 |
475.36 | 3.81 | 3.81 |
615.63 | 6.02 | 6.02 |
551.57 | 4.01 | 4.01 |
555.64 | 8.87 | 8.87 |
502.43 | 5.07 | 5.07 |
515.52 | 4.46 | 4.46 |
539.55 | 3.94 | 3.94 |
476.35 | 3.21 | 3.21 |
595.67 | 4.03 | 4.03 |
566.58 | 4.43 | 4.43 |
436.19 | 3.90 | 3.90 |
527.53 | 4.43 | 4.43 |
651.69 | 5.57 | 5.57 |
589.64 | 3.97 | 3.97 |
516.46 | 5.46 | 5.46 |
697.85 | 9.20 | 9.20 |
797.96 | 10.77 | 10.77 |
412.17 | 4.41 | 4.41 |
557.55 | 3.91 | 3.91 |
563.58 | 3.97 | 3.97 |
739.88 | 9.38 | 9.38 |