Assay Report Card

Basic Information

ID: ALA4192104

Type: Binding

Description: Modulation of human alpha1beta2delta GABAA receptor expressed in Xenopus laevis oocytes assessed as increase in GABA-induced current by measuring rebound current at 1 mM at -60 mV holding potential measured after termination of compound application by two-electrode voltage clamp electrophysiology method relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
308.361.451.45
306.392.092.09
278.331.361.36
306.392.142.14