ID: ALA4194884
Type: Binding
Description: Binding affinity to His-tagged BRD4 bromodomain 1 to 2 (K57 to K550 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by bromodomain TR-FRET binding assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4194884
Ki
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
385.49 | 2.90 | 2.90 |
293.37 | 3.36 | 3.36 |
371.46 | 2.76 | 2.76 |
459.47 | 4.37 | 4.37 |
383.47 | 2.67 | 2.67 |
411.48 | 2.33 | 2.33 |
293.37 | 3.36 | 3.36 |
411.48 | 2.33 | 2.33 |
455.49 | 4.01 | 4.01 |
471.49 | 3.62 | 3.62 |
385.49 | 2.90 | 2.90 |
383.47 | 2.67 | 2.67 |
420.49 | 3.12 | 3.12 |
461.53 | 3.98 | 3.98 |
401.44 | 2.16 | 2.16 |
397.50 | 2.81 | 2.81 |
397.50 | 2.81 | 2.81 |
437.50 | 3.87 | 3.87 |
471.49 | 3.62 | 3.62 |
420.49 | 3.12 | 3.12 |
435.51 | 3.34 | 3.34 |
371.46 | 2.76 | 2.76 |
305.38 | 3.26 | 3.26 |
437.50 | 3.87 | 3.87 |
455.49 | 4.01 | 4.01 |
305.38 | 3.26 | 3.26 |
399.47 | 2.33 | 2.33 |
452.51 | 4.09 | 4.09 |