Basic Information
ID: ALA4200085
Type: Functional
Description: Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of calcium mobilization after 1 hr by Oregon Green BAPTA-1/AM dye-based fluorescence assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Uracil nucleotide/cysteinyl leukotriene receptor(ALA1075162)
Document: ALA4196130
Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of calcium mobilization after 1 hr by Oregon Green BAPTA-1/AM dye-based fluorescence assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4200085
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 233.22 | 1.88 | 1.88 |
| 283.28 | 3.04 | 3.04 |
| 251.21 | 2.02 | 2.02 |
| 325.32 | 3.68 | 3.68 |
| 263.25 | 1.89 | 1.89 |
| 269.20 | 2.16 | 2.16 |
| 251.21 | 2.02 | 2.02 |
| 316.14 | 3.20 | 3.20 |
| 267.67 | 2.54 | 2.54 |
| 267.67 | 2.54 | 2.54 |
| 267.67 | 2.54 | 2.54 |
| 267.67 | 2.54 | 2.54 |
| 316.14 | 3.58 | 3.58 |
| 300.10 | 3.27 | 3.27 |
| 263.25 | 1.89 | 1.89 |
| 261.28 | 2.50 | 2.50 |
| 385.42 | 5.22 | 5.22 |
| 374.18 | 3.14 | 3.14 |
| 309.32 | 3.55 | 3.55 |
| 353.80 | 4.11 | 4.11 |
| 251.21 | 2.02 | 2.02 |
| 327.31 | 3.69 | 3.69 |
| 377.11 | 2.63 | 2.63 |
| 285.66 | 2.68 | 2.68 |
| 327.31 | 3.69 | 3.69 |
| 333.38 | 3.84 | 3.84 |
| 353.80 | 4.11 | 4.11 |
| 395.88 | 5.28 | 5.28 |
| 309.32 | 3.55 | 3.55 |
| 367.83 | 4.50 | 4.50 |
| 258.10 | 3.49 | 3.49 |
| 302.11 | 3.19 | 3.19 |
| 299.28 | 3.14 | 3.14 |
| 333.34 | 3.75 | 3.75 |
| 361.76 | 4.34 | 4.34 |
| 361.76 | 4.34 | 4.34 |
| 330.11 | 2.78 | 2.78 |
| 263.25 | 1.89 | 1.89 |
| 345.30 | 3.83 | 3.83 |
| 302.11 | 3.19 | 3.19 |
| 367.83 | 4.50 | 4.50 |
| 377.11 | 2.63 | 2.63 |
| 302.11 | 3.19 | 3.19 |
| 330.11 | 2.78 | 2.78 |
| 395.88 | 5.28 | 5.28 |
| 330.11 | 2.78 | 2.78 |
| 336.56 | 3.84 | 3.84 |
| 315.35 | 3.61 | 3.61 |
| 317.27 | 3.28 | 3.28 |
| 323.35 | 3.47 | 3.47 |
| 275.30 | 3.01 | 3.01 |