ID: ALA4201837
Type: Binding
Description: Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 assessed as Kinact/Ki ratio pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 mins
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4201837
Ratio
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
416.48 | 4.00 | 4.00 |