Assay Report Card

Basic Information

ID: ALA4201837

Type: Binding

Description: Inhibition of His-6-tagged human KLK6 R74G/R76Q/N132Q mutant expressed in Escherichia coli DH10 assessed as Kinact/Ki ratio pre-incubated for 30 mins before N-Boc-FSR-AMC substrate addition and measured after 30 mins

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
416.484.004.00