Basic Information
ID: ALA4219298
Type: Binding
Description: Induction of cereblon/cullin 4A-mediated BRD2 degradation in human RS4:11 cells at 1 nM after 3 hrs in presence of BET inhibitor 4-((3-Cyclopropyl-1-ethyl-1H-pyrazol-5-yl)amino)-7-(3,5-dimethylisoxazol-4-yl)-6-methoxy-N-methyl-9H-pyrimido[4,5-b]-indole-2-carboxamide by Western blot method
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4219298
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 798.90 | 6.13 | 6.13 |