Basic Information
ID: ALA4219416
Type: Binding
Description: Induction of human His-tagged CRBN-DDB1/GST-tagged BRD4 (49 to 170 residues) interaction assessed as CRBN/DDB1/BRD4/compound ternary complex formation preincubated for 60 mins and measured after 60 mins by luminescence based Alphascreen proximity assay relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4219416
%max
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 457.00 | 5.53 | 5.53 |
| 785.28 | 3.68 | 3.68 |
| 781.25 | 3.58 | 3.58 |
| 869.36 | 3.61 | 3.61 |
| 825.31 | 3.59 | 3.59 |
| 957.47 | 3.64 | 3.64 |
| 913.41 | 3.63 | 3.63 |