Assay Report Card

Basic Information

ID: ALA4219417

Type: Binding

Description: Induction of human His-tagged VHL(1 to 154)/GST-tagged BRD4 (49 to 170 residues) interaction assessed as VHL/BRD4/compound complex formation preincubated for 60 mins and measured after 60 mins by luminescence based Alphascreen proximity assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1039.69
995.635.215.21
1002.66
1171.84
1127.79
1083.74