Basic Information
ID: ALA4219529
Type: Binding
Description: Induction of interaction of N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) co-expressed in Escherichia coli BL21 (DE3) with recombinant human Brd4 BD2 assessed as VCB/BRD4/compound ternary complex formation by isothermal titration calorimetry-based assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4219529
Kd
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1080.75 | ||
| 1002.66 | ||
| 958.61 | 5.58 | 5.58 |
| 1046.71 | ||
| 992.64 | 7.31 | 7.31 |
| 1036.69 |