Assay Report Card

Basic Information

ID: ALA4219618

Type: Binding

Description: Positive allosteric modulation of recombinant human GABAA receptor alpha2beta3gamma2 expressed in CHOK1 cells assessed as potentiation of GABA-induced current at 10 uM at -60 mV holding potential by whole cell patch-clamp method relative to GABA

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
346.382.732.73