Basic Information
ID: ALA4229836
Type: Binding
Description: Displacement of [3H]-8-OH-DPAT from human 5-HT1AR expressed in HEK293 cell membranes after 1 hr by microbeta counting method
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4229836
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 326.83 | 3.72 | 3.72 |
| 375.87 | 4.43 | 4.43 |
| 410.49 | 3.59 | 3.59 |
| 412.95 | 3.81 | 3.81 |
| 312.44 | 3.44 | 3.44 |
| 448.39 | 4.86 | 4.86 |
| 489.65 | 4.08 | 4.08 |
| 508.64 | 3.37 | 3.37 |
| 506.70 | 4.81 | 4.81 |
| 507.69 | 4.21 | 4.21 |
| 493.66 | 3.82 | 3.82 |
| 507.69 | 4.21 | 4.21 |
| 492.67 | 4.42 | 4.42 |
| 506.70 | 4.81 | 4.81 |
| 535.74 | 4.99 | 4.99 |
| 521.71 | 4.60 | 4.60 |
| 507.62 | 3.03 | 3.03 |
| 506.70 | 4.81 | 4.81 |
| 508.62 | 4.94 | 4.94 |
| 521.71 | 4.60 | 4.60 |
| 534.75 | 5.60 | 5.60 |
| 508.64 | 3.37 | 3.37 |
| 489.65 | 4.08 | 4.08 |
| 508.64 | 3.37 | 3.37 |
| 507.69 | 4.21 | 4.21 |
| 507.69 | 4.21 | 4.21 |
| 507.62 | 3.03 | 3.03 |
| 493.66 | 3.82 | 3.82 |
| 491.62 | 3.74 | 3.74 |
| 506.70 | 4.81 | 4.81 |
| 492.67 | 4.42 | 4.42 |
| 520.72 | 5.21 | 5.21 |
| 506.70 | 4.81 | 4.81 |
| 508.62 | 4.94 | 4.94 |
| 534.75 | 5.60 | 5.60 |
| 521.09 | 5.70 | 5.70 |
| 489.65 | 4.08 | 4.08 |
| 507.69 | 4.21 | 4.21 |
| 521.09 | 5.70 | 5.70 |
| 507.69 | 4.21 | 4.21 |
| 507.62 | 3.03 | 3.03 |
| 508.64 | 3.37 | 3.37 |
| 506.70 | 4.81 | 4.81 |
| 520.72 | 5.21 | 5.21 |
| 489.65 | 4.08 | 4.08 |
| 491.62 | 3.74 | 3.74 |
| 521.09 | 5.70 | 5.70 |
| 491.62 | 3.74 | 3.74 |
| 521.09 | 5.70 | 5.70 |
| 535.74 | 4.99 | 4.99 |
| 508.62 | 4.94 | 4.94 |