Basic Information
ID: ALA4233071
Type: Binding
Description: Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate incubated for 10 mins followed by substrate addition measured after 1 hr by spectrofluorimetric method
Format: BAO_0000357
Organism: Homo sapiens
Target: Proteasome Macropain subunit MB1(ALA4662)
Document: ALA4229412
Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate incubated for 10 mins followed by substrate addition measured after 1 hr by spectrofluorimetric method: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4233071
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 384.25 | ||
| 294.12 | ||
| 517.13 | ||
| 361.03 | ||
| 388.32 | ||
| 346.24 | ||
| 272.15 | ||
| 258.13 | ||
| 362.28 | ||
| 334.23 | ||
| 286.18 | ||
| 405.09 | ||
| 256.11 | ||
| 360.26 | ||
| 244.10 | ||
| 376.31 | ||
| 362.28 | ||
| 286.18 | ||
| 474.19 | ||
| 284.17 | ||
| 390.33 | ||
| 272.15 | ||
| 346.24 | ||
| 298.19 | ||
| 338.17 | ||
| 390.29 |