Assay Report Card

Basic Information

ID: ALA4234637

Type: Binding

Description: Activation of full-length recombinant N-terminal His-tagged human AMPKalpha2beta2gamma1 expressed in Escherichia coli BL21 cells at 1 nM using Cy-5 SAMS peptide as substrate preincubated for 60 mins followed by substrate addition and measured after 60 mins in presence of PP2a by TR-FRET assay relative to AMP control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
341.794.564.56
345.793.663.66
357.365.055.05
533.482.402.40
517.921.911.91
521.911.011.01