Assay Report Card

Basic Information

ID: ALA4234770

Type: Binding

Description: Inhibition of Trypanosoma brucei rhodesiense rhodesain assessed as second-order rate constant using Cbz-Phe-Arg-AMC as substrate measured for 30 mins by fluorescence method

Organism: Trypanosoma brucei rhodesiense

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
439.551.661.66
494.593.743.74
516.593.643.64
529.634.194.19
452.512.722.72
521.612.452.45
544.654.124.12
510.633.933.93
494.593.743.74
508.624.134.13
419.522.422.42
454.522.512.51
544.654.124.12
521.612.452.45
605.744.884.88
418.492.522.52
495.623.993.99
487.602.252.25
602.763.233.23
453.542.622.62
523.632.242.24
542.634.334.33