Assay Report Card

Basic Information

ID: ALA4235233

Type: Binding

Description: Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pretreated for 5 mins followed by GSK1016790A addition by Fluo-4-AM dye based fluorescence assay

Organism: Rattus norvegicus

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
316.495.645.64
442.386.066.06
408.637.677.67
316.495.645.64
316.495.645.64
316.495.645.64