Basic Information
ID: ALA4235267
Type: Binding
Description: Antagonist activity at recombinant human ERalpha expressed in HEK293 cells assessed as inhibition of estradiol-induced YFP-fused SRC1 coactivator recruitment measured after 1 hr in presence of Coelenterazine H by BRET assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4235267
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 387.52 | 5.70 | 5.70 |
| 502.66 | 5.92 | 5.92 |
| 518.65 | 5.76 | 5.76 |
| 474.60 | 5.14 | 5.14 |
| 446.55 | 4.82 | 4.82 |