Assay Report Card

Basic Information

ID: ALA4236656

Type: Binding

Description: Irreversible inhibition of BRD4 in human MV4-11 cells assessed as suppression of GRP183 mRNA levels preincubated for 4 hrs followed by compound washout measured after 4 to 24 hrs post washout by RT-PCR analysis

Organism: Homo sapiens

Cell type: MV4-11

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
340.353.383.38