Assay Report Card

Basic Information

ID: ALA4236715

Type: Binding

Description: Non-competitive antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins followed by agonist addition by Fuo-4-AM dependent spectrofluorimetry based Schild analysis

Organism: Rattus norvegicus

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
417.637.057.05
381.656.696.69
667.71