Assay Report Card

Basic Information

ID: ALA4253036

Type: ADME

Description: Inhibition of human 11beta-HSD2 expressed in HEK293 cell lysates at 200 uM using [1,2,6,7-3H]-cortisol as substrate preincubated for 10 mins followed by substrate addition in presence of NAD by scintillation counting relative to control

Organism: Homo sapiens

Subcellular Fraction: Lysate

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
226.282.642.64
294.333.883.88