Assay Report Card

Basic Information

ID: ALA4255286

Type: Functional

Description: Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in forskolin-stimulated cAMP level at 10 uM by BRET assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
476.066.816.81
365.434.014.01
479.575.035.03
465.554.944.94
407.515.105.10
506.645.385.38