Inhibition of [3H]2-m-AzTax binding to P-gp in human SKVLB1 cell plasma membranes assessed as residual [3H]2-m-AzTax binding at 40 uM treated for 30 m...

Basic Information

ID: ALA4255498

Type: Binding

Description: Inhibition of [3H]2-m-AzTax binding to P-gp in human SKVLB1 cell plasma membranes assessed as residual [3H]2-m-AzTax binding at 40 uM treated for 30 mins followed by UV irradiation measured after 10 mins by fluorographic method relative to control

Format: BAO_0000249

Organism: Homo sapiens

Target:  Unchecked(ALA612545)

Document:  ALA4251679

Inhibition of [3H]2-m-AzTax binding to P-gp in human SKVLB1 cell plasma membranes assessed as residual [3H]2-m-AzTax binding at 40 uM treated for 30 mins followed by UV irradiation measured after 10 mins by fluorographic method relative to control: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
853.923.743.74
807.893.263.26
894.934.684.68
853.963.813.81
820.334.594.59