Assay Report Card

Basic Information

ID: ALA4255966

Type: Binding

Description: Inhibition of human His6-tagged BRD4 BD1 (N44 to E168 residues) expressed in Escherichia coli BL21 (DE3) cells using H-SGRGK(Ac)GGK(Ac)GLGK(Ac)GGAK(Ac)RHRK-Biotin-OH as substrate after 2.5 hrs by AlphaScreen assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
457.005.535.53
369.352.272.27
339.402.052.05
384.823.393.39
338.432.872.87
396.853.263.26
298.361.951.95
510.413.973.97
350.372.742.74
346.412.912.91
471.333.383.38
475.754.024.02
347.402.302.30
390.422.382.38
457.303.073.07
338.412.662.66
313.381.731.73
441.303.373.37
384.823.393.39
312.392.342.34
411.283.363.36
484.373.433.43
368.362.882.88
351.362.132.13
526.413.203.20
332.382.602.60